sustanon-250-cycle

Sustanon 250: COURSE

Sustanon or “Sust” is a drug whose composition is represented by several forms of testosterone. Initially Sustanon 250, which was first released by the American company Organon, was used exclusively for therapeutic purposes, was prescribed to patients whose body did not produce the right amount of testosterone. Today this mix has gained wide popularity in sports pharmacology.

Sustanon 250 includes four testosterone esters:

  • Decanoate;
  • Propionate;
  • Isocaproate;
  • Phenylpropionate.

The rate of absorption of each form is different, which explains the high efficacy of the drug. It maintains a high level of testosterone for a whole month. The first to enter the bloodstream is propionate, followed by phenylpropionate, after which isocaproate comes into action, the decanoate is absorbed into the latter.

The duration of action reduces the number of injections. This does not affect the effectiveness of the mixture. It is in no way inferior to drugs that are administered separately. The only drawback is the cost. The mixture, as a rule, is more expensive.

Steroid profile

  • Anabolic and androgenic activity from taking the drug is 100% of testosterone.
  • There is a pronounced suppression of the hypothalamic-pituitary-gonadal system.
  • The mixture has no effect on the liver.
  • The possible detection time in the doping control test is up to three months after the last administration.
  • The drug is given in the form of injections.

Effects on the body

The drug has a multifaceted effect:

Muscle mass is significantly increased. Thanks to the solo course, you can gain about six kilograms.
Strengths increase, and catabolic processes decrease.
Improves endurance, increases the number of red blood cells, activates the processes of hematopoiesis.
Increases sexual desire and libido.
The appetite increases.
Course Sustanon 250 solo
You can start taking this steroid to people who do not have contraindications to the drug that have reached adulthood. Independently the drug is taken for 6-8 weeks. A longer period implies an additional gonadotropin intake. Maintaining an unchanged high concentration of testosterone in the blood requires daily injection. The recommended dosage varies between 250-500 ml.

Aromatase inhibitors start taking from the eighth day of the course and finish after one to two weeks. 21 days after the end of the use, Sustanon 250 begins post-course therapy (PCT) to restore the production of its own testosterone in the body. To the usual mark, the hormone returns about 30 days after the use of boosters. To improve the result allows diet and sports specialized nutrition.

Side effects

Sustanon does not differ from other forms of testosterone, it also shows estrogenic activity. On the background of his admission, the following consequences may occur:

Observed depression of their own hormonal background;
Appear excess fatty deposits;
Develop swelling;
Manifest gynecomastia.
Eliminate these reactions allows timely administration of antiestrogens. The best are aromatase inhibitors. Selective estrogen receptor modulators, including Tamoxifen, begin to be used during the PCT period.

Atrophy of the testicles is the most severe side effect that occurs when taking Sustanon. To prevent its development allows a strictly limited two-month course of injections or parallel use of gonadotropin, as well as the use of antiestrogens.

The instruction to the preparation, as a rule, contains all the necessary information on how to achieve maximum effect and reduce negative manifestations.

Reviews about the drug Sustanon 250

Most negative reviews about the drug are related to the appearance at the injection site of a mixture of seals – infiltrates. This is a temporary phenomenon, which takes place two to five weeks after the end of the course, which is not faced by those who can correctly do injections. There are among the host Sustanon athletes who are unhappy with the effect of fat burning, as together with the muscles often grows and fatty layer.

Strengths from the suspension increase quite well. Athletes who take Sustanon, note the savings of time and money by combining several forms of the hormone and the lack of the need for frequent injections. The price of the drug is not very different from the purchase of aether separately

sustanon

Pharmacodynamics sustanon increases the permeability of the membranes of the cells of helminths for calcium ions, which causes generalized muscle contraction parasites and helminths inhibits glucose uptake by cells, thus reducing glycogen levels and stimulates the release of lactic acid compounds. The result is death of the parasite. sustanon is specifically active against cestodes and trematodes. Pharmacokinetics Absorption.Following oral administration sustanon is rapidly and completely absorbed. Maximum plasma concentration is achieved within 1-2 hours. The half-life of the drug in an unmodified form 1-2.5 hours with metabolites -. 4 hours to achieve a therapeutic effect needed for 4-6 (up to 10) hours to maintain the concentration of drug in the plasma equal to 0.19 mg / l. Distribution. It penetrates through the blood-brain barrier; CSF concentration is 10-20% of the plasma concentration.Penetrates into breast milk at a concentration of 20-25% of the serum concentration. Metabolism. Undergoes metabolism “first pass” through the liver. The main metabolites – hydroxylated products sustanon degradation. Withdrawal. Is carried out mainly through the kidneys. More than 80% of the dose excreted within 4 days, 90% of this amount -. 24 hours Renal failure. Since the drug predominantly renal route of excretion, when renal failure may be slowing down its elimination.Hepatic failure. In decompensated liver failure reduced drug metabolism in the liver, which is accompanied by elongation and increased half-life in the blood concentration of sustanon.

testimony

  • Treatment of infections caused by different types of schistosomes (S. haematobium, S. mansoni, S.intercalatum, S.japonicum, S.mekongi)
  • Treatment of infections caused by liver fluke (Clonorchis sinensis, Opistorchis viverrini) and lung fluke (Paragonimus westermani, et al. Types)

 

Contraindications

  • Hypersensitivity to any component of the drug;
  • Cysticercosis of eye;
  • Interactions with rifampicin.
  • Children under 4 years of age (safety and efficacy not established)

Be wary – decompensated liver failure, gepatolienalny schistosomiasis, cardiac arrhythmia.

 

Application of pregnancy and lactation
biltricid not recommended in the first 3 months of pregnancy. During the short course of therapy biltricid breast-feeding should be suspended for the whole period and the subsequent 24 hours.

Dosage and administration:
The tablet should be taken orally as a whole, without chewing, with a small amount of liquid before or during a meal. If the recommended single dose of the drug per day, the tablet should be taken in the evening. Repeated use of the drug during the day is recommended interval between doses of at least 4 and not more than 6 hours. Adults and children older than 4 years doses biltricid chosen strictly individual and depend on the type of pathogen. By Schistosoma haematobium: 40 mg / kg of body weight once. Duration of treatment 1 day. Schistosoma mansoni and Schistosoma intercalatum: 40 mg / kg 1 time a day or 20 mg / kg two times a day. Duration of treatment 1 day. Schistosoma japonicum, Schistosoma mekongi: 60 mg / kg 1 time a day or 30 mg / kg two times a day. Duration of treatment 1 day.Clonorchis sinensis, Opistorchis viverrini: 25 mg / kg, 3 times a day for 1-3 days. Paragonimus westermani, and other species: 25 mg / kg, 3 times a day for 2-3 days. For children up to 4 years. Safety of the drug in children younger than 4 years have not been established.

Side effects

with the incidence of> 10% Digestive system: abdominal pain, nausea, vomiting. Central nervous system: headache, dizziness. With the incidence of> 1% and <10% Digestive system: lack of appetite.Central nervous system: dizziness, drowsiness. body as a whole: asthenia, fever. Musculoskeletal: myalgia. Skin: . urticaria With incidence of <0.01% body as a whole: allergic reactions (including generalized) including polyserositis. Digestive system: diarrhea mixed with blood. Cardiovascular system: arrhythmia. Central nervous system: convulsions. Adverse reactions can be caused both by sustanon (I, a direct relationship), as result of the endogenous response to the death of the parasite (II, an indirect relationship), and also be symptoms of infection (III, no relation). It is very difficult to make a differential diagnosis between I, II and III of the options and establish the exact cause of adverse reactions.

The interaction with other drugs

While the use of drugs that induce enzyme system of liver cytochrome P450, such as anticonvulsants, dexamethasone concentration sustanon in plasma can be reduced, and in combination with drugs that inhibit these enzymes, such as cimetidine – rise. Chloroquine decreases sustanon concentration in blood plasma.

Cautions
When decompensated liver disease and schistosomiasis gepatolienalny biltricid should be used with caution because of the risk of its longer presence in elevated concentrations in the bloodstream, including collateral vessels. Such patients for treatment may be hospitalized. In cases of cardiac arrhythmias, and while receiving treatment with drugs digitalis biltricid should be carried out under medical supervision.
Patients who live or lived in endemic for cysticercosis and trematodozov areas recommended for treatment in a hospital.

Effects on ability to drive / moving mechanisms
When applying biltricid should refrain from driving / moving mechanisms in the day / day of the drug, and over the next 24 hours.

Form release
On 6 tablets in a bottle amber glass, equipped with a plastic stopper; 1 bottle with instruction on use in a cardboard box shop steroids cheap ephedrine steroidwithdrawal.biz